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- W2024401746 abstract "A series of highly potent and selective inhibitors of DPP-4 was optimized for ADMET properties. The effort resulted in the discovery of inhibitor 1g, that exhibits excellent efficacy in an oral glucose tolerance test and an attractive pharmacokinetic profile." @default.
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- W2024401746 date "2009-08-01" @default.
- W2024401746 modified "2023-10-18" @default.
- W2024401746 title "From lead to preclinical candidate: Optimization of β-homophenylalanine based inhibitors of dipeptidyl peptidase IV" @default.
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- W2024401746 doi "https://doi.org/10.1016/j.bmcl.2009.06.036" @default.
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