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- W2024507493 abstract "Specific3H-1-quinuclidinylbenzilate (3H-1-QNB) binding to rat cochlea homogenates occurs to a homogeneous class of binding sites withKd = 0.13 ± 0.01nMandBmax = 0.57 ± 0.07fmolper cochlea. Binding is stereoselectivity inhibited by benzetimide enantiomers. Dexetimide was more effective than levetimide in displacing3H-1-QNB from its binding sites (Ki = 4 × 10−10Mand 6.5 × 10−6M, respectively). Pirenzepine inhibits3H-1-QNB binding with low affinity (Ki = 2 × 10−6M), classifying the binding sites as muscarinic M2 receptors." @default.
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- W2024507493 date "1988-11-01" @default.
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- W2024507493 title "Cholinergic muscarinic receptors in rat cochlea" @default.
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- W2024507493 doi "https://doi.org/10.1016/0006-8993(88)90682-8" @default.
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