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- W2026228354 abstract "In membranes of neuroblastoma × glioma hybrid (NG108‐15) cells, bradykinin (EC 50 ≅ 5 nM) stimulates GTP hydrolysis by a high‐affinity GTPase ( K m ≅ 0.2 μM). The octapeptide, des‐Arg 9 ‐bradykinin, was inactive. Stimulation of GTP hydrolysis by bradykinin and an opioid agonist was partially additive. Treatment of NG108‐15 cells with pertussis toxin, which inactivates N i , eliminated GTPase stimulation by the opioid agonist but not by bradykinin. The data suggest that bradykinin activates in NG108‐15 membranes a guanine nucleotide‐binding protein which is not sensitive to pertussis toxin and which may be involved in brady‐kinin‐induced stimulation of phosphoinositide metabolism in these cells." @default.
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- W2026228354 date "1986-02-17" @default.
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- W2026228354 title "Bradykinin stimulates GTP hydrolysis in NG108-15 membranes by a high-affinity, pertussis toxin-insensitive GTPase" @default.
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- W2026228354 doi "https://doi.org/10.1016/0014-5793(86)80263-0" @default.
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