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- W2028673022 abstract "The syntheses and structure–activity relationships of the tartrate-based TACE inhibitors are discussed. The optimization of both the prime and non-prime sites led to compounds with picomolar activity. Several analogs demonstrated good rat pharmacokinetics." @default.
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- W2028673022 date "2010-08-01" @default.
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- W2028673022 title "Structure and activity relationships of tartrate-based TACE inhibitors" @default.
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- W2028673022 doi "https://doi.org/10.1016/j.bmcl.2010.06.104" @default.
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