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- W2028852562 abstract "Forty caffeate analogues were synthesized via a convenient method starting from vanillin with moderate to good yields. The testing of biological activity of these compounds against HIV-1 integrase indicates that four compounds: bornyl caffeate, bornyl 2-nitrocaffeate, 5-nitrocaffeic acid and 5-nitrocaffeic acid phenethyl ester (5-nitroCAPE) possess a good HIV integrase inhibitory activity, IC50 19.9, 26.8, 25.0 and 13.5 μM, respectively. Twelve caffeate analogues were tested by MTT assay on growth of human hepatocellular carcinoma BEL-7404, human breast MCF-7 adenocarcinoma, human lung A549 adenocarcinoma and human gastric cancer BCG823 cell lines, respectively. And the best result is IC50 5.5 μM for CAPE against BEL-7404." @default.
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- W2028852562 date "2008-12-01" @default.
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- W2028852562 title "Synthesis of trans-caffeate analogues and their bioactivities against HIV-1 integrase and cancer cell lines" @default.
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- W2028852562 doi "https://doi.org/10.1016/j.bmcl.2008.10.046" @default.
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