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- W2029377926 abstract "Cromakalim, pinacidil and nitroprusside provoked concentration-dependent relaxations of K+-depolarized rat aortae. Glibenclamide, tolbutamide and to a lesser extent tetraethylammonium antagonized the vasorelaxant action of cromakalim and pinacidil. Cromakalim, pinacidil but not nitroprusside elicited a marked increase in 86Rb outflow from preloaded and perifused aortic rings. These increases in 86Rb outflow were inhibited in a concentration-dependent manner by glibenclamide and tetraethylammonium. Our data extend previous observations indicating the involvement of K+ channels in the vasorelaxant properties of cromakalim and pinacidil. Moreover, the present findings suggest that both compounds could interfere with a vascular type of ATP-sensitive K+ channels." @default.
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- W2029377926 title "Hypoglycemic Sulfonylureas Antagonize the Effects of Cromakalim and Pinacidil on <sup>86</sup>Rb Fluxes and Contractile Activity in the Rat Aorta" @default.
- W2029377926 doi "https://doi.org/10.1159/000138697" @default.
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