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- W2032178647 endingPage "91" @default.
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- W2032178647 abstract "Modulators of the arachidonic acid cascade have been in the focus of research for treatments of inflammation and pain for several decades. Targeting this complex pathway experiences a paradigm change towards the design and development of multi-target inhibitors, exhibiting improved efficacy and less undesired side effects. This minireview summarizes recent developments in the field of designed multi-target ligands of the arachidonic acid cascade. In addition to the well-known dual inhibitors of 5-lipoxygenase and cyclooxygenase-2 such as licofelone, very recent developments are discussed. Especially, multi-target inhibitors interfering with the cytochrome P450 pathway via inhibition of soluble epoxide hydrolase seem to offer a novel opportunity for development of novel anti-inflammatory drugs." @default.
- W2032178647 created "2016-06-24" @default.
- W2032178647 creator A5002124394 @default.
- W2032178647 creator A5060739026 @default.
- W2032178647 creator A5082078699 @default.
- W2032178647 date "2013-10-11" @default.
- W2032178647 modified "2023-10-16" @default.
- W2032178647 title "Inhibitors of the Arachidonic Acid Cascade: Interfering with Multiple Pathways" @default.
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- W2032178647 doi "https://doi.org/10.1111/bcpt.12134" @default.
- W2032178647 hasPubMedId "https://pubmed.ncbi.nlm.nih.gov/24015667" @default.
- W2032178647 hasPublicationYear "2013" @default.
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