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- W2032194854 abstract "Tricyclic sulfones were designed as gamma-secretase inhibitors and found to have excellent potency. Extensive SAR shows that a large number of sulfonamides at position 7 of the tricycle are very well tolerated. Compounds such as 15a and 15c showed remarkable in vivo potency." @default.
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- W2032194854 date "2010-06-01" @default.
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- W2032194854 title "Tricyclic sulfones as orally active γ-secretase inhibitors: Synthesis and structure–activity relationship studies" @default.
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- W2032194854 doi "https://doi.org/10.1016/j.bmcl.2010.04.104" @default.
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