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- W2034005177 abstract "A series of fused tricyclic mGluR1 antagonists containing a pyridone ring were synthesized. In vitro, these antagonists were potent against both human and rat isozymes, as well as selective for inhibiting mGluR1 over mGluR5. When dosed orally, several examples were active in vivo in a rat SNL test." @default.
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- W2034005177 date "2012-02-01" @default.
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- W2034005177 title "Fused tricyclic mGluR1 antagonists for the treatment of neuropathic pain" @default.
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- W2034005177 doi "https://doi.org/10.1016/j.bmcl.2011.12.131" @default.
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