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- W2034269403 endingPage "144" @default.
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- W2034269403 abstract "Diseases of the central nervous system present a challenge for the development of new therapeutic agents. Nuclear receptors are ligand-activated transcription factors that have proven to be valuable targets for development of new drugs owing to their ability to directly regulate gene expression. The nuclear receptor, peroxisome proliferator-activated receptor γ (PPARγ), has been investigated for its action in ameliorating the development and progression of a number of CNS diseases. PPARγ agonists exhibit potent anti-inflammatory effects and appear to have direct neuroprotective actions. PPARγ agonists have been shown to be efficacious in animal models of Alzheimer's disease, stroke, multiple sclerosis, Parkinson's disease and amyotrophic lateral sclerosis. The availability of FDA-approved agonists of this receptor will facilitate the rapid translation of these findings into clinical trials for a number of CNS diseases." @default.
- W2034269403 created "2016-06-24" @default.
- W2034269403 creator A5053637497 @default.
- W2034269403 creator A5058419004 @default.
- W2034269403 creator A5073496526 @default.
- W2034269403 creator A5078440867 @default.
- W2034269403 date "2006-07-01" @default.
- W2034269403 modified "2023-10-16" @default.
- W2034269403 title "PPARγ as a therapeutic target in central nervous system diseases" @default.
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- W2034269403 doi "https://doi.org/10.1016/j.neuint.2006.03.020" @default.
- W2034269403 hasPubMedId "https://pubmed.ncbi.nlm.nih.gov/16766086" @default.
- W2034269403 hasPublicationYear "2006" @default.