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- W2034684273 endingPage "440" @default.
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- W2034684273 abstract "Introduction: Anxiety disorders are considered the most common mental disorders and they can increase the risk for comorbid mood and substance use disorders, significantly contributing to the global burden of disease. For this reason, anxiolytics are the most prescribed psychoactive drugs, particularly in the Western world. Areas covered: This review aims to analyze pharmacokinetic profile, plasma level variations so as the metabolism, interactions and possible relation to clinical effect of several drugs which are used primarily as anxiolytics. The drugs analyzed include benzodiazepines, anticonvulsants (pregabalin, gabapentin), buspirone, β-blockers and antihistamines (hydroxyzine). Regarding the most frequently used anxiolytic benzodiazepines, data on alprazolam, bromazepam, chlordesmethyldiazepam, chlordiazepoxide, clotiazepam, diazepam, etizolam, lorazepam, oxazepam, prazepam and clonazepam have been detailed. Expert opinion: There is a need for a more balanced assessment of the benefits and risks associated with benzodiazepine use, particularly considering pharmacokinetic profile of the drugs to ensure that patients, who would truly benefit from these agents, are not denied appropriate treatment. An optimal pharmacological approach involving an integrative pharmacokinetic and pharmacodynamic optimization strategy would ensure better treatment and personalization of anxiety disorders. So it would be desirable for the development of new anxiolytic drug(s) that are more selective, fast acting and free from the unwanted effects associated with the traditional benzodiazepines as tolerance or dependence." @default.
- W2034684273 created "2016-06-24" @default.
- W2034684273 creator A5001736129 @default.
- W2034684273 creator A5013556761 @default.
- W2034684273 creator A5037059287 @default.
- W2034684273 creator A5057104235 @default.
- W2034684273 creator A5069907248 @default.
- W2034684273 creator A5070775561 @default.
- W2034684273 date "2013-01-21" @default.
- W2034684273 modified "2023-09-27" @default.
- W2034684273 title "Understanding the pharmacokinetics of anxiolytic drugs" @default.
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