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- W2035729648 abstract "Histone deacetylase (HDAC) inhibitors are a class of potential therapeutics for the treatment of cancer. Bicyclic tetrapeptides equipped with methoxymethyl ketone and boronic acid as zinc-binding group were designed and synthesized. The inhibitory activities of these compounds were evaluated against HDAC enzymes. The cell-free and cell-based assay data showed that both potency and selectivity changed with the change in zinc-binding group. Boronic acid-based compound showed poor activity whereas methoxymethyl ketone-based compound displayed impressive activity in both cell-free and cell-based conditions." @default.
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- W2035729648 date "2014-12-01" @default.
- W2035729648 modified "2023-09-25" @default.
- W2035729648 title "Bicyclic tetrapeptide histone deacetylase inhibitors with methoxymethyl ketone and boronic acid zinc-binding groups" @default.
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- W2035729648 doi "https://doi.org/10.1016/j.bioorg.2014.10.003" @default.
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