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- W2037852973 endingPage "496" @default.
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- W2037852973 abstract "The mammalian ionotropic glutamate receptor family encodes 18 gene products that coassemble to form ligand-gated ion channels containing an agonist recognition site, a transmembrane ion permeation pathway, and gating elements that couple agonist-induced conformational changes to the opening or closing of the permeation pore. Glutamate receptors mediate fast excitatory synaptic transmission in the central nervous system and are localized on neuronal and non-neuronal cells. These receptors regulate a broad spectrum of processes in the brain, spinal cord, retina, and peripheral nervous system. Glutamate receptors are postulated to play important roles in numerous neurological diseases and have attracted intense scrutiny. The description of glutamate receptor structure, including its transmembrane elements, reveals a complex assembly of multiple semiautonomous extracellular domains linked to a pore-forming element with striking resemblance to an inverted potassium channel. In this review we discuss International Union of Basic and Clinical Pharmacology glutamate receptor nomenclature, structure, assembly, accessory subunits, interacting proteins, gene expression and translation, post-translational modifications, agonist and antagonist pharmacology, allosteric modulation, mechanisms of gating and permeation, roles in normal physiological function, as well as the potential therapeutic use of pharmacological agents acting at glutamate receptors." @default.
- W2037852973 created "2016-06-24" @default.
- W2037852973 creator A5003402513 @default.
- W2037852973 creator A5015251858 @default.
- W2037852973 creator A5017011355 @default.
- W2037852973 creator A5041161550 @default.
- W2037852973 creator A5041248710 @default.
- W2037852973 creator A5058115904 @default.
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- W2037852973 creator A5086505931 @default.
- W2037852973 creator A5087721977 @default.
- W2037852973 creator A5091825209 @default.
- W2037852973 date "2010-08-17" @default.
- W2037852973 modified "2023-10-18" @default.
- W2037852973 title "Glutamate Receptor Ion Channels: Structure, Regulation, and Function" @default.
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