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- W2038585210 abstract "The dimerization and trimerization of the Dmt-Tic, Dmt-Aia and Dmt-Aba pharmacophores provided multiple ligands which were evaluated in vitro for opioid receptor binding and functional activity. Whereas the Tic- and Aba multimers proved to be dual and balanced δ/μ antagonists, as determined by the functional [S35]GTPγS binding assay, the dimerization of potent Aia-based ‘parent’ ligands unexpectedly resulted in substantial less efficient receptor binding and non-active dimeric compounds." @default.
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- W2038585210 date "2010-03-01" @default.
- W2038585210 modified "2023-10-11" @default.
- W2038585210 title "Novel multiple opioid ligands based on 4-aminobenzazepinone (Aba), azepinoindole (Aia) and tetrahydroisoquinoline (Tic) scaffolds" @default.
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- W2038585210 doi "https://doi.org/10.1016/j.bmcl.2010.01.055" @default.
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