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- W2040390015 abstract "A set of cyclic peptide analogues of a selective CXCR4 antagonist FC131 [cyclo(-D-Tyr-Arg-Arg-Nal-Gly-)] were synthesized and bioevaluated. Using (E)-alkene and (Z)-fluoroalkene dipeptide isosteres for Arg-Arg and Arg-Nal substructures, indispensable or the partial contribution of the two peptide bonds to the CXCR4 antagonism and anti-HIV activity was demonstrated. FC131 and the analogues were shown to selectively inhibit SDF-1 binding to CXCR4, whereas no inhibition of binding of SDF-1 to CXCR7 was observed." @default.
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- W2040390015 date "2010-01-01" @default.
- W2040390015 modified "2023-10-18" @default.
- W2040390015 title "Synthesis and biological evaluation of selective CXCR4 antagonists containing alkene dipeptide isosteres" @default.
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- W2040390015 doi "https://doi.org/10.1039/b917236j" @default.
- W2040390015 hasPubMedId "https://pubmed.ncbi.nlm.nih.gov/20090978" @default.
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