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- W2041698840 abstract "Syntheses and pharmacological properties of a new series of acyliminothiadiazoline derivatives 1 are described. These compounds exhibited angiotensin II receptor antagonistic activities in vitro and in vivo. Among them, the compound 1g (KRH-594) showed the strongest antihypertensive action in renal hypertensive rats after oral administration, and its oral bioavailability in dogs was also found to be high (73%)." @default.
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- W2041698840 date "1996-07-01" @default.
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- W2041698840 title "Acyliminothiadiazoline derivatives: New, highly potent, and orally active angiotensin II receptor antagonists" @default.
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- W2041698840 doi "https://doi.org/10.1016/s0960-894x(96)00250-8" @default.
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