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- W2045677482 abstract "To compare the effects of grapefruit juice (GFJ) on the pharmacokinetics of pitavastatin and atorvastatin.In a randomized, four-phase crossover study, eight healthy subjects consumed either GFJ or water t.i.d. for 4 days in each trial. On each final day, a single dose of 4 mg pitavastatin or 20 mg atorvastatin was administered.GFJ increased the mean AUC(0-24) of atorvastatin acid by 83% (95% CI 23-144%) and that of pitavastatin acid by 13% (-3 to 29%).Pitavastatin, unlike atorvastatin, appears to be scarcely affected by the CYP3A4-mediated metabolism." @default.
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- W2045677482 date "2005-11-01" @default.
- W2045677482 modified "2023-10-13" @default.
- W2045677482 title "Effects of grapefruit juice on the pharmacokinetics of pitavastatin and atorvastatin" @default.
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- W2045677482 doi "https://doi.org/10.1111/j.1365-2125.2005.02462.x" @default.
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