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- W204570669 abstract "MicroRNAs (miRNAs) are a class of evolutionally conserved, endogenous, short (18–24 nucleotides), noncoding RNAs that post-transcriptionally downregulate gene expression via translational repression or mRNA degradation. miRNAs regulate every aspect of cellular function, including differentiation, proliferation, and apoptosis. Recently, the roles of miRNAs in the metabolism of xenobiotics and endobiotics were uncovered. Evidence is accumulating that miRNAs regulate the expression of cytochrome P450s, which are major drug-metabolizing enzymes, through direct and/or indirect targeting. Knowledge of pharmacogenetics with respect to drug metabolism has been growing, and miRNA-related single-nucleotide polymorphisms (SNPs) have become a new area of research in this field. The SNPs in miRNA genes or target sites may modify miRNA expression or regulation, thus causing variability in drug response and toxicity. Because miRNAs are differentially expressed in diseases and play critical roles in various biological pathways, they are seen as potential therapeutic targets or a new class of biomarkers. Regulation by miRNAs is a critical factor of inter- and intraindividual variability in drug response and toxicity; thus, miRNAs may be utilized to realize individualized medicine." @default.
- W204570669 created "2016-06-24" @default.
- W204570669 creator A5001851785 @default.
- W204570669 creator A5089297113 @default.
- W204570669 date "2014-01-01" @default.
- W204570669 modified "2023-10-18" @default.
- W204570669 title "MicroRNA: Regulation of P450 and Pharmacogenetics" @default.
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- W204570669 doi "https://doi.org/10.1016/b978-0-12-386882-4.00019-0" @default.
- W204570669 hasPublicationYear "2014" @default.