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- W2047341915 abstract "ヒストン脱アセチル化酵素 (HDAC) は, クロマチンの構造と機能を制御する酵素として化学遺伝学的に発見された. HDACは発がんや腫瘍血管新生に関与し, その阻害剤はがん細胞に細胞周期停止, 分化, アポトーシスなどを誘導することから, 近年, がんの分子標的としての重要性が大変注目されている.本稿では, HDAC阻害剤に関する化学と生物学について, 最近の進歩と今後の展望について述べたい." @default.
- W2047341915 created "2016-06-24" @default.
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- W2047341915 date "2006-01-01" @default.
- W2047341915 modified "2023-09-25" @default.
- W2047341915 title "Drug discovery from chemical genetics on histone deacetylase" @default.
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- W2047341915 doi "https://doi.org/10.2745/dds.21.32" @default.
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