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- W2048397780 endingPage "84" @default.
- W2048397780 startingPage "71" @default.
- W2048397780 abstract "ATP-binding cassette (ABC) genes play a role in the resistance of malignant cells to anticancer agents. The ABC gene products, including ABCB1 (P-glycoprotein), ABCC1 (MRP1), ABCC2 (MRP2, cMOAT), and ABCG2 (BCRP, MXR, ABCP) are also known to influence oral absorption and disposition of a wide variety of drugs. As a result, the expression levels of these proteins in humans have important consequences for an individual's susceptibility to certain drug-induced side effects, interactions, and treatment efficacy. Naturally occurring variants in ABC transporter genes have been identified that might affect the function and expression of the protein. This review focuses on recent advances in the pharmacogenomics of ABC transporters, and discusses potential implications of genetic variants for the chemotherapeutic treatment of cancer." @default.
- W2048397780 created "2016-06-24" @default.
- W2048397780 creator A5001321994 @default.
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- W2048397780 creator A5065279964 @default.
- W2048397780 creator A5079722956 @default.
- W2048397780 creator A5083693387 @default.
- W2048397780 date "2003-04-01" @default.
- W2048397780 modified "2023-10-15" @default.
- W2048397780 title "Pharmacogenomics of ABC transporters and its role in cancer chemotherapy" @default.
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