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• W2048573632 abstract "G-protein-coupled receptor kinase (GRK)-2 and -5 are emerging therapeutic targets for the treatment of cardiovascular disease. In our efforts to discover novel small molecules to inhibit GRK-2 and -5, a class of compound based on 3-(benzo[d]oxazol-2-yl)-5-(1-(piperidin-4-yl)-1H-pyrazol-4-yl)pyridin-2-amine was identified as a novel hit by high throughput screening campaign. Structural modification of parent benzoxazole scaffolds by introducing substituents on phenyl displayed potent inhibitory activities toward GRK-2 and -5." @default.
• W2048573632 created "2016-06-24" @default.
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• W2048573632 date "2013-12-01" @default.
• W2048573632 modified "2023-10-16" @default.
• W2048573632 title "Design and synthesis of novel 3-(benzo[d]oxazol-2-yl)-5-(1-(piperidin-4-yl)-1H-pyrazol-4-yl)pyridin-2-amine derivatives as selective G-protein-coupled receptor kinase-2 and -5 inhibitors" @default.
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• W2048573632 doi "https://doi.org/10.1016/j.bmcl.2013.10.036" @default.
• W2048573632 hasPubMedId "https://pubmed.ncbi.nlm.nih.gov/24210504" @default.
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