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- W2050137519 abstract "The kinin B1 receptors (B1Rs), stimulated by des-Arg9-kinins, are completely inducible, notably following treatment of animals with bacterial lipopolysaccharide. Several studies based on cultured cells have suggested a form of autoregulation of kinin receptors, because B2 receptor (B2R) or B1R stimulation could transcriptionally upregulate B1R expression. The B2R may rather be downregulated in inflammatory conditions. A rabbit B2R-green fluorescent protein (GFP) conjugate stably expressed in HEK 293 cells was rapidly internalized in response to the agonist bradykinin. Ligand-induced receptor cycling was documented applying confocal microscopy. The results confirm agonist-induced B2R endocytosis, but extensive recycling to the cell membrane does not support agonist-induced downregulation." @default.
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- W2050137519 date "2001-01-06" @default.
- W2050137519 modified "2023-09-26" @default.
- W2050137519 title "Ligand-Mediated Regulation of Kinin Receptors in the Rabbit" @default.
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- W2050137519 doi "https://doi.org/10.1515/bc.2001.019" @default.
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