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- W2051069812 abstract "To improve the pharmacokinetics of a previously reported series of dipeptidyl nitrile cathepsin B inhibitors, the P(2)-P(3) amide group was replaced with an arylamine. Further optimization of this template resulted in highly potent and selective inhibitors with excellent oral availability." @default.
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- W2051069812 date "2003-11-01" @default.
- W2051069812 modified "2023-10-03" @default.
- W2051069812 title "N-Arylaminonitriles as bioavailable peptidomimetic inhibitors of cathepsin B" @default.
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- W2051069812 doi "https://doi.org/10.1016/j.bmcl.2003.08.006" @default.
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