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- W2051225174 abstract "Cancer chemotherapy is limited by significant inter-individual variations in responses and toxicities. Such variations are often due to genetic alterations in drug metabolising enzymes (pharmacokinetic polymorphisms) or receptor expression (pharmacodynamic polymorphisms). Pharmacogenetic screening prior to anticancer drug administration may lead to identification of specific populations predisposed to drug toxicity or poor drug responses. The role of polymorphisms in specific enzymes, such as thiopurine S-methyltransferases (TPMT), dihydropyrimidine dehydrogenase (DPD), aldehyde dehydrogenases (ALDH), glutathione S-transferases (GST), uridine diphosphate glucuronosyltransferases (UGTs) and cytochrome P450 (CYP 450) enzymes in cancer therapy are discussed in this review." @default.
- W2051225174 created "2016-06-24" @default.
- W2051225174 creator A5032438481 @default.
- W2051225174 creator A5068268371 @default.
- W2051225174 date "1998-09-01" @default.
- W2051225174 modified "2023-10-17" @default.
- W2051225174 title "Pharmacogenetics and cancer chemotherapy" @default.
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