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- W2051259700 endingPage "380" @default.
- W2051259700 startingPage "371" @default.
- W2051259700 abstract "GABA is a major inhibitory neurotransmitter in the CNS where it regulates neuronal excitability. These actions of GABA are mediated through GABA receptor subtypes, one of which is the GABAB receptor (GBR). The development of specific agonists and antagonists for GBRs has led to a better understanding of their functional roles, which mainly focus on the long-term modulation of neural activity. In this review, the authors emphasize the current knowledge of the structure-action profile of compounds active at GBRs, characterizing their physiology and pharmacology and highlighting their potential as targets for drug development." @default.
- W2051259700 created "2016-06-24" @default.
- W2051259700 creator A5008013016 @default.
- W2051259700 creator A5014641463 @default.
- W2051259700 date "1996-09-01" @default.
- W2051259700 modified "2023-09-23" @default.
- W2051259700 title "GABAB receptors: targets for drug development" @default.
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