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- W2051344554 abstract "Structure–activity relationship on a novel ketone class of H3R antagonists/inverse agonists is disclosed. Compound 4 showed excellent target potency, selectivity and brain penetration. Evaluation of antagonist 4 in the rat EEG/EMG model demonstrated robust wake activity thereby establishing preclinical proof of concept." @default.
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- W2051344554 date "2012-02-01" @default.
- W2051344554 modified "2023-09-26" @default.
- W2051344554 title "Novel morpholine ketone analogs as potent histamine H3 receptor inverse agonists with wake activity" @default.
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- W2051344554 doi "https://doi.org/10.1016/j.bmcl.2012.01.004" @default.
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