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- W2053637598 abstract "Furazolidone (FZ), one of the nitrofuran fungicides, is used as a veterinary medicine in the Middle and Far Eastern countries. In this study, FZ (125 mg/kg) was administered orally to Wistar rats for 3 days. Results of the Ames test using the S-9 fraction of rats treated with FZ showed a significant increase in the number of revertant colonies. Western blot analysis of hepatic CYP isozymes induced by FZ, revealed a remarkable induction of CYP1A1 apoprotein, but CYP1A2 and CYP2E1 apoproteins were not altered. In addition, the expression of CYP1A1 mRNA level in rats treated with FZ by RT-PCR was significantly enhanced by FZ treatment. We concluded that FZ is apparently mutagenic and induces transcription of the CYP1A1 isozyme, which metabolically activates numerous promutagens, in hepatocytes." @default.
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- W2053637598 date "2008-01-01" @default.
- W2053637598 modified "2023-09-24" @default.
- W2053637598 title "Antibiotic Furazolidone Induces CYP1A But Not CYP2E1 Subfamily in Rat Liver" @default.
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- W2053637598 doi "https://doi.org/10.1292/jvms.70.223" @default.
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