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- W2053803797 abstract "Both progesterone receptor modulators (PRMs) as well as pure progesterone antagonists (PAs) have numerous proven and potential therapeutic applications in female health care. Mifepristone, a PRM with only marginal agonistic activity, together with a prostaglandin can terminate pregnancies of less than 9 weeks duration; mifepristone is also used in the preparation of women at later gestational stages whose pregnancies are terminated with prostaglandins or surgery. Mifepristone causes expulsion of the uterine contents following intrauterine fetal death and promotes dilation of the non-pregnant primigravid uterus. It is also effective in the treatment of missed abortion. Together with methotrexate, mifepristone can be used in the medical treatment of ectopic pregnancy. Both PAs and PRMs display antiproliferative effects on the endometrium. Because of this, they have application in the treatment of endometriosis, an estrogen-dependent condition. They may also be utilized to reduce myoma size, acting as both a PA and antiproliferative agent. Unlike GnRH agonists, long-term use in endometriosis and myoma is not associated with loss of bone and hypoestrogenism. PRMs may also be useful in IVF programs to prevent a premature LH surge and to delay the emergence of the implantation window. Some PRMs have potential use as hormone replacement therapy in women during menopause or in those with dysfunctional uterine bleeding." @default.
- W2053803797 created "2016-06-24" @default.
- W2053803797 creator A5024726200 @default.
- W2053803797 creator A5088324465 @default.
- W2053803797 date "2000-11-01" @default.
- W2053803797 modified "2023-10-15" @default.
- W2053803797 title "Progesterone receptor modulators and progesterone antagonists in women's health" @default.
- W2053803797 cites W1463735117 @default.
- W2053803797 cites W1531102169 @default.
- W2053803797 cites W1840935595 @default.
- W2053803797 cites W1840984513 @default.
- W2053803797 cites W1898708016 @default.
- W2053803797 cites W1910306760 @default.
- W2053803797 cites W1911221999 @default.
- W2053803797 cites W1917913033 @default.
- W2053803797 cites W1966828434 @default.
- W2053803797 cites W1967330535 @default.
- W2053803797 cites W1968251168 @default.
- W2053803797 cites W1970539961 @default.
- W2053803797 cites W1971445831 @default.
- W2053803797 cites W1972365601 @default.
- W2053803797 cites W1973830856 @default.
- W2053803797 cites W1974272316 @default.
- W2053803797 cites W1974377866 @default.
- W2053803797 cites W1975486822 @default.
- W2053803797 cites W1976368322 @default.
- W2053803797 cites W1981384075 @default.
- W2053803797 cites W1984862997 @default.
- W2053803797 cites W1987244077 @default.
- W2053803797 cites W1992344390 @default.
- W2053803797 cites W1992512486 @default.
- W2053803797 cites W1992542867 @default.
- W2053803797 cites W2005256844 @default.
- W2053803797 cites W2007951223 @default.
- W2053803797 cites W2012326197 @default.
- W2053803797 cites W2012487133 @default.
- W2053803797 cites W2015742238 @default.
- W2053803797 cites W2016450355 @default.
- W2053803797 cites W2017728147 @default.
- W2053803797 cites W2018398766 @default.
- W2053803797 cites W2023185400 @default.
- W2053803797 cites W2024480273 @default.
- W2053803797 cites W2034215598 @default.
- W2053803797 cites W2038969187 @default.
- W2053803797 cites W2040549856 @default.
- W2053803797 cites W2047203443 @default.
- W2053803797 cites W2047347660 @default.
- W2053803797 cites W2047982918 @default.
- W2053803797 cites W2048924271 @default.
- W2053803797 cites W2048957217 @default.
- W2053803797 cites W2051527207 @default.
- W2053803797 cites W2053688057 @default.
- W2053803797 cites W2056375703 @default.
- W2053803797 cites W2056447394 @default.
- W2053803797 cites W2056834448 @default.
- W2053803797 cites W2057662292 @default.
- W2053803797 cites W2059015734 @default.
- W2053803797 cites W2059587221 @default.
- W2053803797 cites W2061581560 @default.
- W2053803797 cites W2064504572 @default.
- W2053803797 cites W2064960854 @default.
- W2053803797 cites W2068426934 @default.
- W2053803797 cites W2072652930 @default.
- W2053803797 cites W2073187669 @default.
- W2053803797 cites W2076758573 @default.
- W2053803797 cites W2077969055 @default.
- W2053803797 cites W2079241337 @default.
- W2053803797 cites W2082004104 @default.
- W2053803797 cites W2084629480 @default.
- W2053803797 cites W2084815884 @default.
- W2053803797 cites W2089758602 @default.
- W2053803797 cites W2090285649 @default.
- W2053803797 cites W2091156943 @default.
- W2053803797 cites W2091540714 @default.
- W2053803797 cites W2093005645 @default.
- W2053803797 cites W2093512443 @default.
- W2053803797 cites W2094733937 @default.
- W2053803797 cites W2095669679 @default.
- W2053803797 cites W2096662576 @default.
- W2053803797 cites W2099389398 @default.
- W2053803797 cites W2109270155 @default.
- W2053803797 cites W2113737235 @default.
- W2053803797 cites W2117145164 @default.
- W2053803797 cites W2121830948 @default.
- W2053803797 cites W2123015098 @default.
- W2053803797 cites W2125336329 @default.
- W2053803797 cites W2131868790 @default.
- W2053803797 cites W2141790367 @default.
- W2053803797 cites W2163104520 @default.
- W2053803797 cites W2164108954 @default.
- W2053803797 cites W2166686992 @default.
- W2053803797 cites W2170049035 @default.
- W2053803797 cites W2180857759 @default.
- W2053803797 cites W2246590518 @default.
- W2053803797 cites W2261864039 @default.
- W2053803797 cites W2286309563 @default.
- W2053803797 cites W2290286119 @default.
- W2053803797 cites W2294496959 @default.