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- W2055365318 abstract "A novel class of potent and selective alpha-1a receptor antagonists has been identified. The structures of these antagonists were derived from truncating the 4-aryl dihydropyridine subunit present in known alpha-1a antagonists. The design principles which led to the discovery of substituted phenylacetamides, the synthesis and SAR of key analogues, and the results of select in vitro and in vivo studies are described." @default.
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- W2055365318 date "2000-08-01" @default.
- W2055365318 modified "2023-10-14" @default.
- W2055365318 title "Phenylacetamides as selective α-1A adrenergic receptor antagonists" @default.
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- W2055365318 doi "https://doi.org/10.1016/s0960-894x(00)00307-3" @default.
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