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- W2055492722 abstract "An unexpected distribution of the β-adrenergic receptor in the rat lung was revealed by an autoradiographic technique. [3H]-Dihydroalprenolol binding was stereoselective. L-propranolol was 300 times more potent than L-propranolol in competition experiments. Scatchard analysis revealed a Kd of 1.1 nM and Bmax of 14 fmol/mg wet weight. Relative potencies of β-adrenergic ligands were: propranolol > alprenolol > timolol > pindolol > isoproterenol > epinephrine > soterenol > metoprolol > terbutaline > norepinephrine. The autoradiograms generated revealed a diffuse pattern with binding always associated with tissue structures. We conclude that β-adrenergic receptors are extensively distributed in the lung, being present in large and small airways and blood vessels." @default.
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- W2055492722 date "1984-01-01" @default.
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- W2055492722 title "Characterization and Autoradiographic Distribution of the β-Adrenergic Receptor in the Rat Lung" @default.
- W2055492722 doi "https://doi.org/10.1159/000138020" @default.
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