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- W2056521938 abstract "A series of dipeptidyl nitriles as inhibitors of cathepsin K have been explored starting from lead structure 1 (Cbz-Leu-NH-CH2-CN, IC50 = 39 nM). Attachment of non-natural amino acid side chains in P1 and modification of the P3 subunit led to inhibitors with higher potency and improved pharmacokinetic properties." @default.
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- W2056521938 date "2006-05-01" @default.
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- W2056521938 title "Dipeptide nitrile inhibitors of cathepsin K" @default.
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- W2056521938 doi "https://doi.org/10.1016/j.bmcl.2006.01.104" @default.
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