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- W2059430007 abstract "Structural modification of the 2-methoxy group and at the 4-position of the piperidine ring of the 5-HT4 partial agonist 1 led to analogues with increased affinity for the 5-HT4 receptor and loss of agonist activity. Similar modification of 2 resulted in 2-(3,5-dimethoxy) benzyloxy derivatives (23, 24, 26–28) that were found to be 5-HT4 receptor antagonists with subnanomolar affinity." @default.
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- W2059430007 date "1994-10-01" @default.
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- W2059430007 title "Synthesis and preliminary pharmacological evaluation of 2-benzyloxy substituted aryl ketones as 5-HT4 receptor antagonists" @default.
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- W2059430007 doi "https://doi.org/10.1016/s0960-894x(01)80414-5" @default.
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