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- W2060166094 abstract "Two potassium conductances have been isolated in rat Leydig cells by their sensitivity to cytosolic calcium and to K+ channel blockers. We used the whole-cell configuration of the patch-clamp technique to investigate their sensitivity to cyclic AMP, the main messenger of luteinizing hormone, which stimulates Leydig cell steroidogenesis. The voltage-dependent potassium conductance is not modified by exposing the cell to 1 mM chlorophenylthio-cyclic AMP (CPT-cAMP), a membrane-permeant analogue of cAMP. By contrast, the large, calcium-activated potassium conductance is upregulated by CPT-cAMP. Furthermore, the latter is potentiated by the chloride channel blocker 4-acetamido-4'-isothiocyanato-stilbene-2,2'-disulfonic acid, sodium salt (SITS)." @default.
- W2060166094 created "2016-06-24" @default.
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- W2060166094 date "1998-01-01" @default.
- W2060166094 modified "2023-09-25" @default.
- W2060166094 title "Effect of cyclic AMP on the calcium-dependent potassium conductances of rat Leydig cells" @default.
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- W2060166094 doi "https://doi.org/10.1139/cjpp-76-6-649" @default.
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