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- W2060589715 endingPage "2035" @default.
- W2060589715 startingPage "2022" @default.
- W2060589715 abstract "Abstract Since its discovery in the late 1980s, phosphoinositide 3‐kinase (PI3K), and its isoforms have arguably reached the forefront of signal transduction research. Regulation of this lipid kinase, its functions, its effectors, in short its entire signaling network, has been extensively studied. PI3K inhibitors are frequently used in biochemistry and cell biology. In addition, many pharmaceutical companies have launched drug‐discovery programs to identify modulators of PI3Ks. Despite these efforts and a fairly good knowledge of the PI3K signaling network, we still have only a rudimentary picture of the signaling dynamics of PI3K and its lipid products in space and time. It is therefore essential to create and use novel biological and chemical tools to manipulate the phosphoinositide signaling network with spatial and temporal resolution. In this review, we discuss the current and potential future tools that are available and necessary to unravel the various functions of PI3K and its isoforms." @default.
- W2060589715 created "2016-06-24" @default.
- W2060589715 creator A5022080003 @default.
- W2060589715 creator A5069111179 @default.
- W2060589715 date "2012-09-10" @default.
- W2060589715 modified "2023-10-17" @default.
- W2060589715 title "The Chemical Biology of Phosphoinositide 3-Kinases" @default.
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