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- W2061009085 abstract "Resume Pemetrexed est un nouvel antimetabolite multicible, intervenant dans le cycle des folates, mecanisme metabolique indispensable a la synthese de l’ADN. Cet antifolate multicible, contrairement aux antifolates classiques (methotrexate, raltitrexed et lometrexol), inhibe les trois enzymes cles : la Thymidilate Synthetase (TS), la Dihydrofolate Reductase (DHFR) et la GlycinAmide Ribonucleotide FormylTransferase (GARFT). Son activite va dependre de sa penetration a l’interieur de la cellule grâce a differents systemes de transport ainsi que de sa polyglutamation." @default.
- W2061009085 created "2016-06-24" @default.
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- W2061009085 date "2009-06-01" @default.
- W2061009085 modified "2023-09-25" @default.
- W2061009085 title "Les grandes étapes de la personnalisation des traitements en oncologie : spécificité du mode d’action du pemetrexed" @default.
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- W2061009085 doi "https://doi.org/10.1016/s1877-1203(09)75252-8" @default.
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