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- W2062973172 abstract "The novel imidazo[4,5-c]pyridine 1,2,5-oxadiazol-3-yl template affords an excellent start point for identification of inhibitors of a number of protein kinases. Here we report on its optimisation for mitogen and stress-activated protein kinase-1 (MSK-1) inhibitory activity, and selectivity over other kinases." @default.
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- W2062973172 date "2005-07-01" @default.
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- W2062973172 title "(1H-Imidazo[4,5-c]pyridin-2-yl)-1,2,5-oxadiazol-3-ylamine derivatives: Further optimisation as highly potent and selective MSK-1-inhibitors" @default.
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- W2062973172 doi "https://doi.org/10.1016/j.bmcl.2005.05.020" @default.
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