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- W2064865177 abstract "A novel series of pyrrolopyrazole-based protein kinase C β II inhibitors has been identified from high-throughput screening. Herein, we report our initial structure-activity relationship studies with a focus on optimizing compound ligand efficiency and physicochemical properties, which has led to potent inhibitors with good cell permeability." @default.
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- W2064865177 date "2011-01-01" @default.
- W2064865177 modified "2023-10-17" @default.
- W2064865177 title "Identification of novel pyrrolopyrazoles as protein kinase C β II inhibitors" @default.
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- W2064865177 doi "https://doi.org/10.1016/j.bmcl.2010.10.032" @default.
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