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- W2065346882 abstract "It has been demonstrated that once-a-day dosing of systemically-distributed SCD inhibitors leads to adverse events in eye and skin. Herein, we describe our efforts to convert a novel class of systemically-distributed potent triazole-based uHTS hits into liver-targeted SCD inhibitors as a means to circumvent chronic toxicity." @default.
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- W2065346882 date "2011-11-01" @default.
- W2065346882 modified "2023-09-24" @default.
- W2065346882 title "Conversion of systemically-distributed triazole-based stearoyl-CoA desaturase (SCD) uHTS hits into liver-targeted SCD inhibitors" @default.
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- W2065346882 doi "https://doi.org/10.1016/j.bmcl.2011.08.073" @default.
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