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- W2066699098 abstract "Non-small cell lung cancers (NSCLC) harboring anaplastic lymphoma kinase (ALK) gene rearrangements invariably develop resistance to 2nd-generation ALK inhibitors. Lorlatinib (PF-06463922) (6) is a 3rd-generation macrocyclic ALK-TKI that demonstrates many advantages over 2nd-generation ALK inhibitors. Lorlatinib has demonstrated decent kinase selectivity, promising pharmacokinetic profile, selective brain-penetration and strong antiproliferative activity in several ALK/ROS1-driven tumor models. The current review describes the activity spectrum, key events from discovery to clinical applications and the evidences that lorlatinib acts as an ALK/ROS1 inhibitor in clinical settings." @default.
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- W2066699098 date "1999-02-01" @default.
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- W2066699098 title "Involvement of protein tyrosine phosphorylation in immunotoxin effects on T lymphocytes" @default.
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- W2066699098 doi "https://doi.org/10.1016/s0041-1345(98)01766-7" @default.
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