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- W2068179023 endingPage "1180" @default.
- W2068179023 startingPage "1161" @default.
- W2068179023 abstract "The current anti-HIV treatments fail to completely eradicate the virus in HIV-infected individuals, mainly as a result of a small pool of latently infected cells. This issue, together with the emergence of multidrug-resistant viruses, clearly highlights the need to find additional strategies. An overview of the Tat-mediated transcription inhibitors 6-desfluoroquinolones (6-DFQs), identified by our group, is given in this review along with a critical appraisal of their advantages and drawbacks. Attempts are also made to place them within the context of new potential anti-HIV therapeutics. Due to their innovative mechanism of action, the 6-DFQs could be interesting candidates for use in association with the currently used cocktail of drugs. Their potential as antivirals deserves further investigation." @default.
- W2068179023 created "2016-06-24" @default.
- W2068179023 creator A5010835490 @default.
- W2068179023 creator A5043864360 @default.
- W2068179023 creator A5054053277 @default.
- W2068179023 date "2010-07-01" @default.
- W2068179023 modified "2023-10-16" @default.
- W2068179023 title "6-desfluoroquinolones as HIV-1 Tat-mediated transcription inhibitors" @default.
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