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- W2069717129 abstract "Poly(ethylene imine)s (PEIs) are widely used in different applications, but most extensively investigated as non-viral vector systems. The high ability of cationic PEIs to complex and condense negatively charged DNA and RNA combined with their inherent proton sponge behavior accounts for the excellent efficiency in gene delivery. Further chemical modifications of the polymer expand the application potential, primarily aiming at increased transfection efficiency, cell selectivity and reduced cytotoxicity. Improvements in the synthesis of tailor-made PEIs in combination with new in-depth analytical techniques offer the possibility to produce highly purified polymers with defined structures. The contemporary strategies towards linear and branched poly(ethylene imine)s with modified surface characteristics, PEI-based copolymers as well as conjugates with bioactive molecules will be discussed. In this regard, the versatile branched PEIs have been successfully modified in a statistical manner, whereas the linear counterparts open avenues to design and synthesize well-defined architectures, in order to exploit their high potential in gene delivery." @default.
- W2069717129 created "2016-06-24" @default.
- W2069717129 creator A5007304580 @default.
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- W2069717129 creator A5034341324 @default.
- W2069717129 creator A5071910582 @default.
- W2069717129 creator A5075012306 @default.
- W2069717129 date "2012-01-01" @default.
- W2069717129 modified "2023-10-12" @default.
- W2069717129 title "Branched and linear poly(ethylene imine)-based conjugates: synthetic modification, characterization, and application" @default.
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