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- W2069936729 abstract "The characteristics of beta-adrenergic receptors in human fetal lung were examined using the beta-adrenoceptor antagonist 3H-dihydroalprenolol /DHA/. Steady-state binding was reached by 15 min at 25°C, and the association and dissociation rate constants were 0.0422 nM−1 min−1 and 0.0874 min−1, respectively. From saturation experiments, Bmax of 82.0 ± 38 fmol/mg protein and KD=1.85 ± 0.92 nM were calculated. Inhibition of 3H-DNA binding by beta-1 /metoprolol/ and beta-2 /zinterol, IPS-339, fenoterol/ selective drugs resulted in biphasic displacement curves with slope factors less than 1.0. Analysis of these curves revealed a beta-1: beta-2 ratio of 40:60 in human fetal lung. The presence of 3H-DHA binding sites in early human lung may have a developmental importance which is not yet understood." @default.
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- W2069936729 date "1986-03-01" @default.
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- W2069936729 title "Binding properties of beta-adrenergic receptors in early human fetal lung" @default.
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- W2069936729 doi "https://doi.org/10.1016/0006-291x(86)91001-6" @default.
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