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- W2074407377 abstract "An efficient solid-phase synthesis of benzisothiazolone-1,1-dioxide-based serine protease inhibitors involving alkylation of carboxylic acids with N-(bromomethyl)benzisothiazolone-1,1-dioxide has been developed. An example using this procedure for preparation of a library of human mast cell tryptase inhibitors is described." @default.
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- W2074407377 date "1999-03-01" @default.
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- W2074407377 title "Solid-phase synthesis of benzisothiazolones as serine protease inhibitors" @default.
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- W2074407377 doi "https://doi.org/10.1016/s0960-894x(99)00078-5" @default.
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