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• W2076089188 abstract "A series of tricyclic cannabinoids incorporating a heteroaroyl group at C3 were prepared as probes to explore the binding site(s) of the CB1 and CB2 receptors. This relatively unexplored structural motif is shown to be CB2 selective with Ki values at low nanomolar concentrations when the heteroaromatic group is 3-benzothiophenyl (41) or 3-indolyl (50). When photoactivated, the lead compound 41 was shown to successfully label the CB2 receptor through covalent attachment at the active site while 50 failed to label. The benzothiophenone moiety may be a photoactivatable moiety suitable for selective labeling." @default.
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• W2076089188 date "2012-08-01" @default.
• W2076089188 modified "2023-10-01" @default.
• W2076089188 title "C3-Heteroaroyl cannabinoids as photolabeling ligands for the CB2 cannabinoid receptor" @default.
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• W2076089188 doi "https://doi.org/10.1016/j.bmcl.2012.06.013" @default.
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