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- W2076310588 abstract "During efforts to improve the bioavailability of FMS kinase inhibitors 1 and 2, a series of saturated and aromatic 4-heterocycles of reduced basicity were prepared and evaluated in an attempt to also improve the cardiovascular safety profile over lead arylamide 1, which possessed ion channel activity. The resultant compounds retained excellent potency and exhibited diminished ion channel activity." @default.
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- W2076310588 date "2010-07-01" @default.
- W2076310588 modified "2023-10-18" @default.
- W2076310588 title "Reducing ion channel activity in a series of 4-heterocyclic arylamide FMS inhibitors" @default.
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- W2076310588 doi "https://doi.org/10.1016/j.bmcl.2010.05.013" @default.
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