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- W2077373139 endingPage "237" @default.
- W2077373139 startingPage "217" @default.
- W2077373139 abstract "Somatostatin is a peptide with a multitude of functions in the central nervous system and the periphery. It mediates its actions by binding to high-affinity G-protein coupled receptors, genes for five of which (sst1-sst5) have recently been cloned. The somatostatin sst2 receptor exists as two splice variants, sst2(a) and sst2(b) receptors, which differ in length and composition of their intracellular carboxy-termini. In this review, we describe the localisation of the two receptor isoforms in the central nervous system, the periphery and also in tumour tissue. Furthermore, we summarise and discuss the data on the functional properties of the recombinant splice variants that have been generated so far, which include activation of extracellular acidification rates, inhibition of adenylate cyclase and activation of MAP-kinases as well as the transcription factor Elk-1." @default.
- W2077373139 created "2016-06-24" @default.
- W2077373139 creator A5080462590 @default.
- W2077373139 creator A5083627175 @default.
- W2077373139 date "2000-10-01" @default.
- W2077373139 modified "2023-09-26" @default.
- W2077373139 title "Characterisation of somatostatin sst2 receptor splice variants" @default.
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- W2077373139 doi "https://doi.org/10.1016/s0928-4257(00)00207-2" @default.