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- W2078277622 endingPage "836" @default.
- W2078277622 startingPage "822" @default.
- W2078277622 abstract "Of the human solid cancers, Non-Small Cell Lung Cancer (NSCLC) and Malignant Pleural Mesothelioma (MPM) display a natural history supporting the concept that they develop from multiple preneoplastic pathways. Recently, new evidence suggested that nicotinic Acetylcholine Receptors (nAChRs) play a significant role in lung cancer predisposition and natural history. This review is based on some translational research aimed at evaluating the potential therapeutic effect of nAChR antagonists on NSCLC and MPM. The background and rationale of this approach are based on the experimental observations that: (a) NSCLC and MPM cells express nAChRs and (b) the activation of these receptors by agonists, namely nicotine, inhibits apoptosis, whereas receptor antagonists have a pro-apoptotic effect." @default.
- W2078277622 created "2016-06-24" @default.
- W2078277622 creator A5006970882 @default.
- W2078277622 creator A5049337449 @default.
- W2078277622 creator A5055878606 @default.
- W2078277622 creator A5078111994 @default.
- W2078277622 date "2009-09-01" @default.
- W2078277622 modified "2023-10-03" @default.
- W2078277622 title "α7-Nicotinic receptor antagonists at the beginning of a clinical era for NSCLC and Mesothelioma?" @default.
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