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- W2078592807 abstract "An SAR study around the mixed 5-HT1ABD receptor antagonist SB-272183 found that introduction of cis-2,6-dimethyl substitution onto the piperazine ring was a key structural change, which imparted a combination of both excellent selectivity over the 5-HT1A and 5-HT1D receptors and low intrinsic activity. This led to the identification of the selective 5-HT1B receptor antagonist SB-616234." @default.
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- W2078592807 date "2005-11-01" @default.
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- W2078592807 title "Identification of a potent and selective 5-HT1B receptor antagonist" @default.
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