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- W2078657788 abstract "A paramount role in carcinogenesis is played by the tumour-suppressor protein p53. In the case of DNA damage, it leads to cell-cycle arrest or apoptosis. p53 activity is often reduced due to the overexpression of its main regulator, the Mdm2 protein. The discovery of small molecules, such as 1, that are able to inhibit the interaction between p53 and Mdm2 opens up new possibilities for the therapy of malignant diseases." @default.
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- W2078657788 date "2004-11-03" @default.
- W2078657788 modified "2023-09-26" @default.
- W2078657788 title "Novel Activators of the Tumour Suppressor p53" @default.
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- W2078657788 doi "https://doi.org/10.1002/cbic.200400194" @default.
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