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- W2079172002 abstract "Following the description of the [3H]deltorphin II, it has been reported that the modification of deltorphin II with the substitution of Val5,6 residues by the more hydrophobic lle5,6 residues leads to an increased affinity and selectivity. The lle5,6deltorphin II (Tyr-D-Ala-Phe-Gly-lle-lle-Gly-NH2) was tritiated by catalytic dehalogenation and labelled rat brain membrane sites with a Kd value of 0.40 nM and a Bmax of 121 fmol/mg protein. Competition binding experiments with various unlabelled subtype specific opioid receptor ligands resulted in μδ and κδ selectivity ratios of 2400 and 18 000 respectively. Due to its high δ receptor affinity, δ selectivity and very low non-specific binding (<20%), [3H]lle5,6deltorphin II, is a very useful tool for the identification and characterisation of δ opioid receptors." @default.
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- W2079172002 date "1994-04-01" @default.
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- W2079172002 title "Binding characteristics of the novel highly selective delta agonist, [3H]Ile5,6deltorphin II" @default.
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- W2079172002 doi "https://doi.org/10.1016/0143-4179(94)90080-9" @default.
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